Tocris公司代理生物计划 Tocris离子通道调控剂,Tocris/CMPD101/5642/10/10 mg,白蛋白,天然蛋白,蛋白类,,Tocris Bioscience蚂蚁淘商城

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Tocris/CMPD101/5642/10/10 mg

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Tocris

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5642/10

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4000-520-616

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Description:PotentandselectiveGRK2/3inhibitor

ChemicalName:3-[[[4-Methyl-5-(4-pyridinyl)-4H-1,2,4-triazol-3-yl]methyl]amino]-N-[[2-(trifluoromethyl)phenyl]methyl]benzamide

Purity:≥98%(HPLC)

BIOLOGicalActivityTechnicalDataSolubilityCalculatorsDatasheetsReferences

BiologicalActivity

PotentandselectiveGRK2/3inhibitor(IC₅₀valuesare32and54nMforGRK3andGRK2,respectively).ExhibitsselectivityforGRK2/3overGRK1/5.ReducesDAMGO-induceddesensitizationandinternalizationofμ-opioidreceptors.

TechnicalData

M.Wt	466.46
Formula	C₂₄H₂₁F₃N₆O
Storage	Storeat-20°C
Purity	≥98%(HPLC)
CASNumber	865608-11-3
PubChemID	11677079
InChIKey	WFOVEDJTASPCIR-UHFFFAOYSA-N
Smiles	CN1C(CNC2=CC(C(NCC3=CC=CC=C3C(F)(F)F)=O)=CC=C2)=NN=C1C4=CC=NC=C4

Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.

AllTocrisproductsareintendedforlaboratoryresearchuseonly.

SolubilityData

	Solvent	MaxConc.mg/mL	MaxConc.mM
Solubility
	DMSO	46.65	100
	ethanol	46.65	100

PreparingStockSolutions

Thefollowingdataisbasedontheproductmolecularweight466.46.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.

Concentration/SolventVolume/Mass	1mg	5mg	10mg
1mM	2.14mL	10.72mL	21.44mL
5mM	0.43mL	2.14mL	4.29mL
10mM	0.21mL	1.07mL	2.14mL
50mM	0.04mL	0.21mL	0.43mL

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