Overview:
Potent and selective Src family kinase inhibitor. Inhibits Lck (IC50=4 nM), Fyn (IC50=5 nM), and Hck (IC50=5 nM).Shows weaker inhibition of EGFR (IC50=480 nM) and no inhibition of ZAP-70 (IC50=100 uM) and JAK2 (IC50=50 uM). Useful for probing the involvement of Src family tyrosine kinases in cellular signaling.
References:
1. F. Carlomagno et al.; J. Clin. Endocrinol. Metab. 2003 8:1897 2. J.K. Chen et al.; J Biol Chem. 2000275:13789 3. M. Yoshizumi et al.; J. Biol. Chem. 2000275:11706 4. J.H. Hanke et al.; J. Biol. Chem. 1996271:695
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那糖酵解中依赖NAD的酶不是要在线粒体内反应?
蛋白酶分布广泛,主要存在于人和动物消化道中,而消化道通过口与肛门与外界相通,属于外环境或外界环境
(溶菌酶、凝血酶原等)分布在内环境
(消化)酶分布在消化道

