Thalidomideanalog.Immunemodulatorydrugandcereblonbindingcompound.Inducesubiquitinationanddegradationofcaseinkinase(CK)1αbytheE3ubiquitinligaseCRL4CRBN.AlsoTNF-αinhibitorandangiogenesisinhibitor.
Application
Cereblonbinder;inducesubiquitinationanddegradationofCK1αbyE3ubiquitinligase
ProductInformation
Purity: >97%
MW: 259.26
Formula: C13H13N3O3
CASNumber 191732-72-6
PhysicalState: Lyophilizedwhitetoyellowsolid
Quantity: 1g;5g
Solubility: 25mg/mLinDMSO
Storage: RoomTemperature
Documents
References
1. Petzold etal (2016)Structuralbasisoflenalidomide-inducedCK1adegradationbytheCRL4(CRBN)ubiquitinligase.Nature 532 127PMID: 26909574
2. Krönke etal (2015)LenalidomideinducesubiquitinationanddegradationofCK1αindel(5q)MDS.Nature 523183PMID: 26131937
ebiomall.com
>
>
>
>
>
>
>
>
>
>
>
>
那糖酵解中依赖NAD的酶不是要在线粒体内反应?
蛋白酶分布广泛,主要存在于人和动物消化道中,而消化道通过口与肛门与外界相通,属于外环境或外界环境
(溶菌酶、凝血酶原等)分布在内环境
(消化)酶分布在消化道

