FunctionalizedcereblonligandforPROTACresearchanddevelopment;incorporatesanE3ligaseligandplusashortalkyllinkerreadyforconjugationtoatargetproteinligand.PartofarangeoffunctionalizedtoolmoleculesforPROTACR&D.
Application
FunctionalizedcereblonligandforPROTACs;incorporatesanE3ligaseligandplusashortalkyllinker
ProductInformation
Purity: >95%
MW: 438.86
Formula: C19H22N4O6.HCl
PhysicalState: Lyophilizedwhitesolid
Quantity: 5mg;10mg;25mg
Solubility: 40mg/mLinDMSO;40mg/mLinwater
Storage: Storeat-20C.
References
1. Winter etal (2015)FunctionalizedCereblonligandforPROTACs;incorporatesanE3ligaseligandandalinkerusedinPROTACtechnology.Science 348 1376PMID: 25999370
2. Salami etal (2017)Wastedisposal-Anattractivestrategyforcancertherapy.Science 355 1163PMID: 28302825
Documents
ebiomall.com
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那糖酵解中依赖NAD的酶不是要在线粒体内反应?
蛋白酶分布广泛,主要存在于人和动物消化道中,而消化道通过口与肛门与外界相通,属于外环境或外界环境
(溶菌酶、凝血酶原等)分布在内环境
(消化)酶分布在消化道

