Tocris型号参数规格 Tocris Bioscience授权代理商，正品,Tocris/Aliskiren hemifumarate/5491/50/50 mg,蛋白酶类,Tocris,Bio-Techne,,50 mg蚂蚁淘商城

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Tocris/Aliskiren hemifumarate/5491/50/50 mg

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Tocris/Aliskiren hemifumarate/5491/50/50 mg

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Tocris

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5491/50

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4000-520-616

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Description:Potentrenininhibitor;antihypertensive

AlternativeNames:SPP100

ChemicalName:(αS,γS,δS,ζS)-δ-Amino-N-(3-amino-2,2-dimethyl-3-oxopropyl)-γ-hydroxy-4-methoxy-3-(3-methoxypropoxy)-α,ζ-bis(1-methylethyl)benzeneoctanamidehemifumarate

Purity:≥99%(HPLC)

BIOLOGicalActivityTechnicalDataSolubilityCalculatorsDatasheetsReferences

BiologicalActivity

Potentrenininhibitor(IC₅₀=0.6and80nMforhumanandratrespectively).Exhibitsselectivityforreninoverarangeofotherasparticproteinases(>5000nM).Lowersbloodpressureinahypertensiverodentmodel.Orallyactive.

CompoundLibraries

AliskirenhemifumarateisalsoofferedaspartoftheTocriscreenPlusandTocriscreenLibraryofFDA-ApprovedCompounds.FindoutmoreaboutcompoundlibrariesavailablefromTocris.

TechnicalData

M.Wt	609.83
Formula	C₃₀H₅₃N₃O6.1/2C₄H₄O₄
Storage	Storeat-20°C
Purity	≥99%(HPLC)
CASNumber	173334-58-2
PubChemID	6918427
InChIKey	KLRSDBSKUSSCGU-KRQUFFFQSA-N
Smiles	COC1=C(OCCCOC)C=C(C[C@H]([C@@H](C)C)C[C@@H]([C@@H](O)C[C@@H]([C@@H](C)C)C(NCC(C)(C)C(N)=O)=O)N)C=C1.COC2=C(OCCCOC)C=C(C[C@H]([C@@H](C)C)C[C@@H]([C@@H](O)C[C@@H]([C@@H](C)C)C(NCC(C)(C)C(N)=O)=O)N)C=C2.O=C(/C=C/C(O)=O)O

Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.

AllTocrisproductsareintendedforlaboratoryresearchuseonly.

SolubilityData

	Solvent	MaxConc.mg/mL	MaxConc.mM
Solubility
	DMSO	60.98	100
	water	60.98	100

PreparingStockSolutions

Thefollowingdataisbasedontheproductmolecularweight609.83.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.

Concentration/SolventVolume/Mass	1mg	5mg	10mg
1mM	1.64mL	8.2mL	16.4mL
5mM	0.33mL	1.64mL	3.28mL
10mM	0.16mL	0.82mL	1.64mL
50mM	0.03mL	0.16mL	0.33mL

ProductDatasheets

CertificateofAnalysis/ProductDatasheet

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BiologicalActivity

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