BiologicalActivity
Subtilisin/Kex2p-likeproproteinconvertaseinhibitor;blocksactivityofallsevenconvertases(PC1,PC2,PC4,PACE4,PC5,PC7andfurin).AbolishesproET-1processinginendothelialcells;inhibitsregulatedsecretionoftheneuronalpolypeptideVGFinPC12cells.
TechnicalData
| M.Wt | 744.42 |
| Formula | C34H66ClN11O5 |
| Sequence | RVKR (Modifications:Arg-1=Decanoyl-Arg,Arg-4=chlororomethylketone) |
| Storage | Storeat-20°C |
| CASNumber | 150113-99-8 |
| PubChemID | 9962075 |
| InChIKey | NHBJTTGFHCHQHS-VZTVMPNDSA-N |
| Smiles | [H]N([C@@H](CCCNC(N)=N)C(=O)N[C@@H](C(C)C)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(N)=N)C(=O)CCl)C(=O)CCCCCCCCC |
Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.
AllTocrisproductsareintendedforlaboratoryresearchuseonly.
SolubilityData
| Solubility | Solubleto1mg/mlinwater |
PreparingStockSolutions
Thefollowingdataisbasedontheproductmolecularweight744.42.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.
| Concentration/SolventVolume/Mass | 1mg | 5mg | 10mg |
|---|---|---|---|
| 1mM | 1.34mL | 6.72mL | 13.43mL |
| 5mM | 0.27mL | 1.34mL | 2.69mL |
| 10mM | 0.13mL | 0.67mL | 1.34mL |
| 50mM | 0.03mL | 0.13mL | 0.27mL |
MolarityCalculator
ReconstitutionCalculator
DilutionCalculator
ProductDatasheets
© 2005- 苏州蚂蚁淘生物科技有限公司 版权所有。
苏ICP备17049038号-11
苏公网安备 32059002001627号
声明：本网站部分产品受外界条件影响（包含但不限于进口国出口国政策限制等因素），无法提供销售服务，下单后，会由客服人员联系厂家确认后另行通知。部分危险品无法清关，请勿下单
我要提问
您的问题将推送给已购用户，TA们将会为你解答。