BiologicalActivity
Highlypotent5-HT1Breceptoragonist(Kivaluesare28,150and1490nMat5-HT1B,5-HT1Aand5-HT2receptorsrespectively).DecreasescentralSEROtoninsynthesisandattenuatesaggressivebehaviorinvivo.Alsoactsasanantagonistat5-HT3receptors(Ki=29.5nM)andisbrainpenetrant.
CompoundLibraries
AnpirtolinehydrochlorideisalsoofferedaspartoftheTocriscreenPlus.FindoutmoreaboutcompoundlibrariesavailablefromTocris.
TechnicalData
| M.Wt | 265.2 |
| Formula | C10H13ClN2S.HCl |
| Storage | Desiccateat+4°C |
| Purity | ≥99%(HPLC) |
| CASNumber | 99201-87-3 |
| PubChemID | 6917943 |
| InChIKey | GRXDJABVNGUGCW-UHFFFAOYSA-N |
| Smiles | Cl.ClC1=NC(SC2CCNCC2)=CC=C1 |
Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.
AllTocrisproductsareintendedforlaboratoryresearchuseonly.
SolubilityData
| Solvent | MaxConc.mg/mL | MaxConc.mM | |
|---|---|---|---|
| Solubility | |||
| DMSO | 26.52 | 100 | |
| water | 100 |
PreparingStockSolutions
Thefollowingdataisbasedontheproductmolecularweight265.2.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.
| Concentration/SolventVolume/Mass | 1mg | 5mg | 10mg |
|---|---|---|---|
| 1mM | 3.77mL | 18.85mL | 37.71mL |
| 5mM | 0.75mL | 3.77mL | 7.54mL |
| 10mM | 0.38mL | 1.89mL | 3.77mL |
| 50mM | 0.08mL | 0.38mL | 0.75mL |
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