BiologicalActivity
Potentandselectiveμopioidreceptorantagonist(Kivaluesare0.96and>10,000nMforμandδreceptorsrespectively).Causesbehavioraleffectsoncentraladministrationinvivo.AlsoincreasesK+currentsinratlocusceruleusneuronsinvitroviaaμreceptorindependentmechanism.
TechnicalData
| M.Wt | 1062.28 |
| Formula | C50H67N11O11S2 |
| Sequence | FCYWXTXT (Modifications:Phe-1=D-Phe,Trp-4=D-Trp,X-5=Orn,X-7=Pen,Disulfidebridgebetween2-7,Thr-8=C-terminalamide) |
| Storage | Desiccateat-20°C |
| CASNumber | 103429-31-8 |
| PubChemID | 90479805 |
| InChIKey | PZWWYAHWHHNCHO-KOFBULAQSA-N |
| Smiles | [H]N[C@H](CC1=CC=CC=C1)C(=O)N[C@H]1CSSC(C)(C)C(NC(=O)[C@@H](NC(=O)[C@H](CCCN)NC(=O)[C@@H](CC2=CNC3=C2C=CC=C3)NC(=O)[C@H](CC2=CC=C(O)C=C2)NC1=O)[C@@H](C)O)C(=O)N[C@@H]([C@@H](C)O)C(N)=O |
Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.
AllTocrisproductsareintendedforlaboratoryresearchuseonly.
SolubilityData
| Solubility | Solubleto1mg/mlinwater |
PreparingStockSolutions
Thefollowingdataisbasedontheproductmolecularweight1062.28.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.
| Concentration/SolventVolume/Mass | 1mg | 5mg | 10mg |
|---|---|---|---|
| 1mM | 0.94mL | 4.71mL | 9.41mL |
| 5mM | 0.19mL | 0.94mL | 1.88mL |
| 10mM | 0.09mL | 0.47mL | 0.94mL |
| 50mM | 0.02mL | 0.09mL | 0.19mL |
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