BiologicalActivity
Non-selective5HT2antagonist,migraineprophylactic.AlsoSETD7/9inhibitor(IC50=1μM).Decreasesexpressionandincreasesdegradationofestrogenreceptor(ER)αinbreasttumorMCF7cells.InhibitsgrowthofMCF7xenograftsinmice.
TechnicalData
| M.Wt | 323.86 |
| Formula | C21H21N.HCl |
| Storage | StoreatRT |
| Purity | ≥98%(HPLC) |
| CASNumber | 969-33-5 |
| PubChemID | 13770 |
| InChIKey | ZPMVNZLARAEGHB-UHFFFAOYSA-N |
| Smiles | Cl[H].CN1CCC(CC1)=C1/C2=C(C=CC=C2)C=CC2=C1C=CC=C2 |
Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.
AllTocrisproductsareintendedforlaboratoryresearchuseonly.
SolubilityData
| Solvent | MaxConc.mg/mL | MaxConc.mM | |
|---|---|---|---|
| Solubility | |||
| DMSO | 32.39 | 100 |
PreparingStockSolutions
Thefollowingdataisbasedontheproductmolecularweight323.86.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.
| Concentration/SolventVolume/Mass | 1mg | 5mg | 10mg |
|---|---|---|---|
| 1mM | 3.09mL | 15.44mL | 30.88mL |
| 5mM | 0.62mL | 3.09mL | 6.18mL |
| 10mM | 0.31mL | 1.54mL | 3.09mL |
| 50mM | 0.06mL | 0.31mL | 0.62mL |
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