BiologicalActivity
PotentERβagonist;displays>200-foldselectivityforERβoverERα(IC50valuesare5and1216nMforhumanERβandERα;3.1and620nMforratERβandERα;and3.7and750nMformouseERβandERαrespectively).
LicensingInformation
SoldforresearchpurposesunderagreementfromPfizerInc.
TechnicalData
| M.Wt | 271.24 |
| Formula | C15H10FNO3 |
| Storage | Storeat-20°C |
| Purity | ≥99%(HPLC) |
| CASNumber | 524684-52-4 |
| PubChemID | 5326893 |
| InChIKey | FCXYSEXZEGPLGG-DHDCSXOGSA-N |
| Smiles | C=CC1=C2C(N=C(C3=CC=C(O)C(F)=C3)O2)=CC(O)=C1 |
Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.
AllTocrisproductsareintendedforlaboratoryresearchuseonly.
SolubilityData
| Solvent | MaxConc.mg/mL | MaxConc.mM | |
|---|---|---|---|
| Solubility | |||
| DMSO | 27.12 | 100 | |
| ethanol | 27.12 | 100 |
PreparingStockSolutions
Thefollowingdataisbasedontheproductmolecularweight271.24.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.
| Concentration/SolventVolume/Mass | 1mg | 5mg | 10mg |
|---|---|---|---|
| 1mM | 3.69mL | 18.43mL | 36.87mL |
| 5mM | 0.74mL | 3.69mL | 7.37mL |
| 10mM | 0.37mL | 1.84mL | 3.69mL |
| 50mM | 0.07mL | 0.37mL | 0.74mL |
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