BiologicalActivity
Verypotentligandforα1sites(Kifordisplacementofprazosin=0.2nM).Displaysdifferentbindingpropertiesforeachα1subtype(pKivaluesare8.74,9.44and9.57forα1B,α1Dandα1Aadrenoceptorsrespectively).Alsobindsto5-HT1Asites(Ki=50nM).
TechnicalData
| M.Wt | 419.48 |
| Formula | C23H25N5O3 |
| Storage | StoreatRT |
| CASNumber | 133399-65-2 |
| PubChemID | 4013695 |
| InChIKey | AQASGOHUMGAWJJ-UHFFFAOYSA-N |
| Smiles | COC1=C(C=CC=C1)N1CCN(CCN2C(=O)NC3=C(NC4=CC=CC=C34)C2=O)CC1 |
Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.
AllTocrisproductsareintendedforlaboratoryresearchuseonly.
SolubilityData
| Solvent | MaxConc.mg/mL | MaxConc.mM | |
|---|---|---|---|
| Solubility | |||
| DMSO | 4.19 | 10mMwithgentlewarming |
PreparingStockSolutions
Thefollowingdataisbasedontheproductmolecularweight419.48.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.
| Concentration/SolventVolume/Mass | 1mg | 5mg | 10mg |
|---|---|---|---|
| 1mM | 2.38mL | 11.92mL | 23.84mL |
| 5mM | 0.48mL | 2.38mL | 4.77mL |
| 10mM | 0.24mL | 1.19mL | 2.38mL |
| 50mM | 0.05mL | 0.24mL | 0.48mL |
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