BiologicalActivity
CB2receptoragonist.Displays4-foldhigheraffinityforthehumanCB2receptorthanthehumanCB1receptor(Kivaluesare43.3and162.4nMrespectively);shows70-foldaffinityfortheratCB2receptorovertheratCB1receptor(Kivaluesare16.3and1130nMrespectively).Attenuatestactileallodyniainaratmodel;doesnotaffectratlocomotoractivity.
TechnicalData
| M.Wt | 349.43 |
| Formula | C21H23N3O2 |
| Storage | Storeat+4°C |
| Purity | ≥99%(HPLC) |
| CASNumber | 1048973-47-2 |
| PubChemID | 25034599 |
| InChIKey | ZGQHMZCITJHYOW-QOCHGBHMSA-N |
| Smiles | O=C(C3=CC=CC=C3)NN=C(C1=CC=CC=C1N2CCCCCC)/C2=O |
Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.
AllTocrisproductsareintendedforlaboratoryresearchuseonly.
SolubilityData
| Solvent | MaxConc.mg/mL | MaxConc.mM | |
|---|---|---|---|
| Solubility | |||
| DMSO | 17.47 | 50 | |
| ethanol | 17.47 | 50 |
PreparingStockSolutions
Thefollowingdataisbasedontheproductmolecularweight349.43.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.
| Concentration/SolventVolume/Mass | 1mg | 5mg | 10mg |
|---|---|---|---|
| 1mM | 2.86mL | 14.31mL | 28.62mL |
| 5mM | 0.57mL | 2.86mL | 5.72mL |
| 10mM | 0.29mL | 1.43mL | 2.86mL |
| 50mM | 0.06mL | 0.29mL | 0.57mL |
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