BiologicalActivity
PotentendogenouscannABInoidandvanilloidreceptoragonist,withnoactionatdopaminereceptors.SelectiveforCB1overCB2receptors(Kivaluesare0.25and12μMrespectively),andpotentagonistatTRPV1(VR1)receptors(EC50~50nM).MetabolicallystableandcompetitivelyinhibitsFAAHandanandamidetransport.Hascannabinoidandvanilloidactionsinvivo.
TechnicalData
| M.Wt | 439.64 |
| Formula | C28H41NO3 |
| Storage | Desiccateat-20°C |
| CASNumber | 199875-69-9 |
| PubChemID | 5282105 |
| InChIKey | MVVPIAAVGAWJNQ-DOFZRALJSA-N |
| Smiles | O=C(NCCC1=CC=C(O)C(O)=C1)CCCC=C/CC=C/C/C=CC/C=CCCCCC |
Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.
AllTocrisproductsareintendedforlaboratoryresearchuseonly.
SolubilityData
| Solubility | Solubleinethanol(suppliedpre-dissolvedinanhydrousethanol,5mg/ml) |
PreparingStockSolutions
Thefollowingdataisbasedontheproductmolecularweight439.64.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.
| Concentration/SolventVolume/Mass | 1mg | 5mg | 10mg |
|---|---|---|---|
| 1mM | 2.27mL | 11.37mL | 22.75mL |
| 5mM | 0.45mL | 2.27mL | 4.55mL |
| 10mM | 0.23mL | 1.14mL | 2.27mL |
| 50mM | 0.05mL | 0.23mL | 0.45mL |
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