BiologicalActivity
PotentandselectiveGPR139agonist(EC50=16nM).SelectiveforGPR139overapanelofGPCRs,ionchannelsandtransporters,includingGPR142.Brainandcellpenetrant.Orallybioavailable.
TechnicalData
| M.Wt | 316.78 |
| Formula | C17H17ClN2O2 |
| Storage | StoreatRT |
| Purity | ≥98%(HPLC) |
| CASNumber | 1802326-66-4 |
| PubChemID | 2548547 |
| InChIKey | MWDVCHRYCKXEBY-LBPRGKRZSA-N |
| Smiles | O=C(CNC(C1=CC=CC(Cl)=C1)=O)N[C@@H](C)C2=CC=CC=C2 |
Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.
AllTocrisproductsareintendedforlaboratoryresearchuseonly.
SolubilityData
| Solvent | MaxConc.mg/mL | MaxConc.mM | |
|---|---|---|---|
| Solubility | |||
| DMSO | 31.68 | 100 | |
| ethanol | 6.34 | 20 |
PreparingStockSolutions
Thefollowingdataisbasedontheproductmolecularweight316.78.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.
| Concentration/SolventVolume/Mass | 1mg | 5mg | 10mg |
|---|---|---|---|
| 1mM | 3.16mL | 15.78mL | 31.57mL |
| 5mM | 0.63mL | 3.16mL | 6.31mL |
| 10mM | 0.32mL | 1.58mL | 3.16mL |
| 50mM | 0.06mL | 0.32mL | 0.63mL |
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