BiologicalActivity
SelectiveadenosineA1receptorantagonist;displays890-foldselectivityforratA1receptorsoverA2Areceptors(Kivaluesare0.19and170nMrespectively).DisplaysnoeffectonrecombinantratA3receptorsexpressedonCHOcellsatconcentrationsupto10μM.Exhibitsdiureticandrenalprotectiveeffectsinrats.
CompoundLibraries
KW3902isalsoofferedaspartoftheTocriscreenPlus.FindoutmoreaboutcompoundlibrariesavailablefromTocris.
TechnicalData
| M.Wt | 356.46 |
| Formula | C20H28N4O2 |
| Storage | Storeat+4°C |
| Purity | ≥99%(HPLC) |
| CASNumber | 136199-02-5 |
| PubChemID | 64627 |
| InChIKey | PJBFVWGQFLYWCB-UHFFFAOYSA-N |
| Smiles | O=C1C2=C(NC(C34CC(CC4C5)CC5C3)=N2)N(CCC)C(N1CCC)=O |
Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.
AllTocrisproductsareintendedforlaboratoryresearchuseonly.
SolubilityData
| Solvent | MaxConc.mg/mL | MaxConc.mM | |
|---|---|---|---|
| Solubility | |||
| DMSO | 17.82 | 50 | |
| ethanol | 8.91 | 25 |
PreparingStockSolutions
Thefollowingdataisbasedontheproductmolecularweight356.46.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.
| Concentration/SolventVolume/Mass | 1mg | 5mg | 10mg |
|---|---|---|---|
| 1mM | 2.81mL | 14.03mL | 28.05mL |
| 5mM | 0.56mL | 2.81mL | 5.61mL |
| 10mM | 0.28mL | 1.4mL | 2.81mL |
| 50mM | 0.06mL | 0.28mL | 0.56mL |
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