BiologicalActivity
Highaffinityμ-opioidreceptoragonistwithperipheralselectivity(Kivaluesare2,48and1156nMforμ-,δ-andκ-opioidreceptorsrespectively).Antidiarrhoealandantihyperalgesicagent.AlsoaCa2+channelblocker;atlowmicromolarconcentrationsitblocksbroadspectrumneuronalHVACa2+channelsandathigherconcentrationsitreducesCa2+fluxthroughNMDAreceptoroperatedchannels.
TechnicalData
| M.Wt | 513.51 |
| Formula | C29H33ClN2O2.HCl |
| Storage | StoreatRT |
| Purity | ≥99%(HPLC) |
| CASNumber | 34552-83-5 |
| PubChemID | 71420 |
| InChIKey | PGYPOBZJRVSMDS-UHFFFAOYSA-N |
| Smiles | Cl.CN(C)C(=O)C(CCN1CCC(O)(CC1)C1=CC=C(Cl)C=C1)(C1=CC=CC=C1)C1=CC=CC=C1 |
Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.
AllTocrisproductsareintendedforlaboratoryresearchuseonly.
SolubilityData
| Solvent | MaxConc.mg/mL | MaxConc.mM | |
|---|---|---|---|
| Solubility | |||
| DMSO | 10.27 | 20 | |
| ethanol | 10.27 | 20 |
PreparingStockSolutions
Thefollowingdataisbasedontheproductmolecularweight513.51.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.
| Concentration/SolventVolume/Mass | 1mg | 5mg | 10mg |
|---|---|---|---|
| 1mM | 1.95mL | 9.74mL | 19.47mL |
| 5mM | 0.39mL | 1.95mL | 3.89mL |
| 10mM | 0.19mL | 0.97mL | 1.95mL |
| 50mM | 0.04mL | 0.19mL | 0.39mL |
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