Tocris试剂产品信息美国Tocris Bioscience公司,Tocris/MA 2029/4934/10/10 mg,受体,生物分子,生化试剂,,Tocris Bioscience蚂蚁淘商城

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Tocris/MA 2029/4934/10/10 mg

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Tocris

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4934/10

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Description:Potentandselective,competitivemotilinreceptorantagoNIST;orallyactive

ChemicalName:4-Fluoro-N-methyl-L-phenylalanyl-N-methyl-L-valyl-3-(1,1-dimethylethyl)-N-ethyl-L-tyrosinamide

Purity:≥98%(HPLC)

BIOLOGicalActivityTechnicalDataSolubilityCalculatorsDatasheetsReferences

BiologicalActivity

Potentandselective,competitivemotilinreceptorantagonist(IC₅₀=4.9nM).Selectiveforthemotilinreceptoroverarangeofotherreceptorsandionchannels.Inhibitsmotilin-inducedduodenalmusclecontractionsinvitro.Alsoinhibitsmotilin-inducedcolonicandaBDominalcontractionsinvivo.Orallyactive.

TechnicalData

M.Wt	556.71
Formula	C₃₁H₄₅FN₄O₄
Storage	Storeat+4°C
Purity	≥98%(HPLC)
CASNumber	287206-61-5
PubChemID	10144175
InChIKey	KSDWAJPUTRBIRR-KLJDGLGGSA-N
Smiles	FC1=CC=C(C[C@H](NC)C(N(C)[C@@H]([C@H](C)C)C(N[C@@H](CC2=CC=C(O)C(C(C)(C)C)=C2)[C@@](NCC)=O)=O)=O)C=C1

Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.

AllTocrisproductsareintendedforlaboratoryresearchuseonly.

SolubilityData

	Solvent	MaxConc.mg/mL	MaxConc.mM
Solubility
	1eq.HCl	11.13	20
	DMSO	55.67	100

PreparingStockSolutions

Thefollowingdataisbasedontheproductmolecularweight556.71.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.

Concentration/SolventVolume/Mass	1mg	5mg	10mg
1mM	1.8mL	8.98mL	17.96mL
5mM	0.36mL	1.8mL	3.59mL
10mM	0.18mL	0.9mL	1.8mL
50mM	0.04mL	0.18mL	0.36mL

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