BiologicalActivity
HighlypotentandselectiveantagonistoftheplateletP2Y1receptor(Ki=0.78nM).InhibitsADP-inducedaggregationofhumanplateletswithanIC50valueof0.95nM.InhibitstheupregulationofNTPDase1byATPγS.Preventsthrombusformationinvivo.
LicensingInformation
SoldunderlicensefromtheNIH,USPatent10/169975
TechnicalData
| M.Wt | 629.29 |
| Formula | C13H18N5O8P2I.4NH3 |
| Storage | Storeat-20°C |
| Purity | ≥96%(HPLC) |
| CASNumber | 630103-23-0 |
| PubChemID | 90488745 |
| InChIKey | FVTFHHDVLNQSME-AVAGOIHISA-N |
| Smiles | IC4=NC1=C(C(NC)=N4)N=CN1[C@H]2C[C@H](OP(O)(O)=O)[C@@]3(COP(O)(O)=O)[C@@H]2C3.N.N.N.N |
Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.
AllTocrisproductsareintendedforlaboratoryresearchuseonly.
SolubilityData
| Solvent | MaxConc.mg/mL | MaxConc.mM | |
|---|---|---|---|
| Solubility | |||
| water | 56.12 | 100 |
PreparingStockSolutions
Thefollowingdataisbasedontheproductmolecularweight629.29.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.
| Concentration/SolventVolume/Mass | 1mg | 5mg | 10mg |
|---|---|---|---|
| 1mM | 1.59mL | 7.95mL | 15.89mL |
| 5mM | 0.32mL | 1.59mL | 3.18mL |
| 10mM | 0.16mL | 0.79mL | 1.59mL |
| 50mM | 0.03mL | 0.16mL | 0.32mL |
MolarityCalculator
ReconstitutionCalculator
DilutionCalculator
ProductDatasheets
© 2005- 苏州蚂蚁淘生物科技有限公司 版权所有。
苏ICP备17049038号-11
苏公网安备 32059002001627号
声明：本网站部分产品受外界条件影响（包含但不限于进口国出口国政策限制等因素），无法提供销售服务，下单后，会由客服人员联系厂家确认后另行通知。部分危险品无法清关，请勿下单
我要提问
您的问题将推送给已购用户，TA们将会为你解答。