BiologicalActivity
Potentandselective5-HT2Cagonist(IC50valuesare12and633nMfor5-HT2Cand5-HT2Areceptorsrespectively).Displayshighaffinityforthe5-HT2Breceptor(Ki=38nM)butactsasaninverseagonist.Activeinvivo;inhibitsscratchinginamousemodelofOCD.
TechnicalData
| M.Wt | 218.29 |
| Formula | C13H18N2O |
| Storage | Storeat+4°C |
| Purity | ≥99%(HPLC) |
| CASNumber | 1465-16-3 |
| PubChemID | 44404883 |
| InChIKey | MZZRFEIDRWKTKJ-UHFFFAOYSA-N |
| Smiles | OC1=C2C(N(C)C=C2CCN(C)C)=CC=C1 |
Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.
AllTocrisproductsareintendedforlaboratoryresearchuseonly.
SolubilityData
| Solvent | MaxConc.mg/mL | MaxConc.mM | |
|---|---|---|---|
| Solubility | |||
| DMSO | 21.83 | 100 | |
| ethanol | 2.18 | 10 |
PreparingStockSolutions
Thefollowingdataisbasedontheproductmolecularweight218.29.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.
| Concentration/SolventVolume/Mass | 1mg | 5mg | 10mg |
|---|---|---|---|
| 1mM | 4.58mL | 22.91mL | 45.81mL |
| 5mM | 0.92mL | 4.58mL | 9.16mL |
| 10mM | 0.46mL | 2.29mL | 4.58mL |
| 50mM | 0.09mL | 0.46mL | 0.92mL |
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