BiologicalActivity
PotentandselectiveneuropeptideYY5receptorantagonist(IC50valuesare3.1,>10000,>10000and>10000nMforY5,Y1,Y2andY4receptorsrespectively).DoesnotblockNPY-inducedfeedinginvivo.Orallyactiveandbrainpenetrant.
CompoundLibraries
NPY5RA972isalsoofferedaspartoftheTocriscreenPlus.FindoutmoreaboutcompoundlibrariesavailablefromTocris.
TechnicalData
| M.Wt | 351.44 |
| Formula | C21H25N3O2 |
| Storage | StoreatRT |
| Purity | ≥98%(HPLC) |
| CASNumber | 439861-56-0 |
| PubChemID | 9884833 |
| InChIKey | ZNFMHLDBJPAFEQ-UHFFFAOYSA-N |
| Smiles | CC1=C(NC(N4CCOCC4)=O)C=CC3=C1C2=CC=CC=C2N3C(C)C |
Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.
AllTocrisproductsareintendedforlaboratoryresearchuseonly.
SolubilityData
| Solvent | MaxConc.mg/mL | MaxConc.mM | |
|---|---|---|---|
| Solubility | |||
| DMSO | 35.14 | 100 |
PreparingStockSolutions
Thefollowingdataisbasedontheproductmolecularweight351.44.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.
| Concentration/SolventVolume/Mass | 1mg | 5mg | 10mg |
|---|---|---|---|
| 1mM | 2.85mL | 14.23mL | 28.45mL |
| 5mM | 0.57mL | 2.85mL | 5.69mL |
| 10mM | 0.28mL | 1.42mL | 2.85mL |
| 50mM | 0.06mL | 0.28mL | 0.57mL |
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