进口Tocris现货 Tocris抗体,Tocris/PD 135158/2608/50/50 mg,受体,生物分子,生化试剂,,Tocris Bioscience蚂蚁淘商城

商品信息

联系客服

郑重提醒：

无质量问题不接受退换货，下单前请仔细核对信息。

下单后请及时联系客服核对商品价格，订单生效后再付款。

Tocris/PD 135158/2608/50/50 mg

品牌 /

Tocris

货号 /

2608/50

官网地址

美元价：

登录查看

(友情提示：该价格仅为参考，欢迎联系客服询价！)

数量：

免费咨询热线

4000-520-616

商品介绍售后保障相关文章商品咨询

联系客服

Description:PotentandselectiveCCK₂antagoNIST

AlternativeNames:CAM1028

ChemicalName:4-[[(1R)-2-[[(2R)-3-(1H-Indol-3-yl)-2-methyl-1-oxo-2-[[[[(1S,2R,4S)-1,7,7-trimethylbicyclo[2.2.1]hept-2-yl]oxy]carbonyl]amino]propyl]amino]-1-phenylethyl]amino]-4-oxobutanoicacid

Purity:≥98%(HPLC)

BIOLOGicalActivityTechnicalDataSolubilityCalculatorsDatasheetsReferences

BiologicalActivity

Potentandselective,nonpeptideCCK₂receptorantagonist(IC₅₀valuesare2.8and1232nMforCCK₂andCCK₁respectively)thatdisplaysnegligIBLeaffinityatGABA_A,benzodiazepine,substanceP,neurotensin,opioid,bradykininand5-HT₃receptors(IC₅₀>10μM).Exhibitsanxiolyticactivityinelevatedplusmazeandsocialinteractiontestsandincreasesfoodintakeinrats.

TechnicalData

M.Wt	616.76
Formula	C₃₅H₄₄N₄O₆
Storage	Storeat+4°C
Purity	≥98%(HPLC)
CASNumber	130285-87-9
PubChemID	44385784
InChIKey	NNTPEWZUKRSTMM-CFHPNWNBSA-N
Smiles	C[C@](NC(OC3C4(C)CCC(C(C)4C)C3)=O)(C(NC[C@@H]([C@]5=CC=CC=C5)NC(CCC(O)=O)=O)=O)CC2=CNC1=CC=CC=C12

Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.

AllTocrisproductsareintendedforlaboratoryresearchuseonly.

SolubilityData

	Solvent	MaxConc.mg/mL	MaxConc.mM
Solubility
Solubility	DMSO	61.68	100

PreparingStockSolutions

Thefollowingdataisbasedontheproductmolecularweight616.76.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.

Concentration/SolventVolume/Mass	1mg	5mg	10mg
1mM	1.62mL	8.11mL	16.21mL
5mM	0.32mL	1.62mL	3.24mL
10mM	0.16mL	0.81mL	1.62mL
50mM	0.03mL	0.16mL	0.32mL

ProductDatasheets

CertificateofAnalysis/ProductDatasheet

SafetyDatasheet

Selectanotherlanguage:

BiologicalActivity

TechnicalData

SolubilityData

PreparingStockSolutions

MolarityCalculator

ReconstitutionCalculator

DilutionCalculator

ProductDatasheets