BiologicalActivity
Selectiveμopioidreceptoragonist(IC50valuesare5.5and>10000nMforinhibitionof125I-FK33,824and125I-DADLEbindingtoμandδsitesrespectively).Producesnaloxone-reversIBLeanalgesia,catalepsyandhyperthermiafollowingcentraladministrationinratsinvivo.
TechnicalData
| M.Wt | 535.64 |
| Formula | C29H37N5O5 |
| Sequence | YPFP (Modifications:Phe-3=N-methyl-Phe,Pro-4=C-terminalamide) |
| Storage | Storeat-20°C |
| CASNumber | 83397-56-2 |
| PubChemID | 10437173 |
| InChIKey | JAKBYSTWCHUQOK-QORCZRPOSA-N |
| Smiles | [H]N[C@@H](CC1=CC=C(O)C=C1)C(=O)N1CCC[C@H]1C(=O)N(C)[C@@H](CC1=CC=CC=C1)C(=O)N1CCC[C@H]1C(N)=O |
Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.
AllTocrisproductsareintendedforlaboratoryresearchuseonly.
SolubilityData
| Solubility | Solubleto1mg/mlinwater |
PreparingStockSolutions
Thefollowingdataisbasedontheproductmolecularweight535.64.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.
| Concentration/SolventVolume/Mass | 1mg | 5mg | 10mg |
|---|---|---|---|
| 1mM | 1.87mL | 9.33mL | 18.67mL |
| 5mM | 0.37mL | 1.87mL | 3.73mL |
| 10mM | 0.19mL | 0.93mL | 1.87mL |
| 50mM | 0.04mL | 0.19mL | 0.37mL |
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