BiologicalActivity
Potent,selective5-HT2receptorantagonist;displayssomeselectivityfor5-HT2Areceptors(Ki=1.6nM).IC50valuesare2.2,310,2400,3700,>5000and>5000nMfor5-HT2,α1-adrenergic,D2dopamine,5-HT1,5-HT3andβ-adrenergicreceptorsrespectively.Inhibits5-HT-inducedplateletaggregationandpressorresponsesinvivo.
CompoundLibraries
R-96544hydrochlorideisalsoofferedaspartoftheTocriscreenPlus.FindoutmoreaboutcompoundlibrariesavailablefromTocris.
TechnicalData
| M.Wt | 391.94 |
| Formula | C22H29NO3.HCl |
| Storage | StoreatRT |
| Purity | ≥99%(HPLC) |
| CASNumber | 167144-80-1 |
| PubChemID | 10668210 |
| InChIKey | OUKRSTJUAQEATQ-GZJHNZOKSA-N |
| Smiles | Cl[H].COC1=CC=CC(CCC2=C(OCC[C@@H]3C[C@@H](O)CN3C)C=CC=C2)=C1 |
Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.
AllTocrisproductsareintendedforlaboratoryresearchuseonly.
SolubilityData
| Solvent | MaxConc.mg/mL | MaxConc.mM | |
|---|---|---|---|
| Solubility | |||
| DMSO | 39.19 | 100 | |
| water | 39.19 | 100 |
PreparingStockSolutions
Thefollowingdataisbasedontheproductmolecularweight391.94.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.
| Concentration/SolventVolume/Mass | 1mg | 5mg | 10mg |
|---|---|---|---|
| 1mM | 2.55mL | 12.76mL | 25.51mL |
| 5mM | 0.51mL | 2.55mL | 5.1mL |
| 10mM | 0.26mL | 1.28mL | 2.55mL |
| 50mM | 0.05mL | 0.26mL | 0.51mL |
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