BiologicalActivity
α1A-adrenoceptorantagonist,withveryhighaffinityforα1Areceptors(pKiandpA2estimatesof9.1-9.9)anda30-100foldselectivityovertheα1Bandα1Dsubtypes(pKiandpA2estimates7.7-7.8).
LicensingInformation
SoldwiththepermissionofRocheBioscience
CompoundLibraries
RS17053hydrochlorideisalsoofferedaspartoftheTocriscreenPlus.FindoutmoreaboutcompoundlibrariesavailablefromTocris.
TechnicalData
| M.Wt | 449.42 |
| Formula | C24H29N2O2Cl.HCl |
| Storage | StoreatRT |
| CASNumber | 169505-93-5 |
| PubChemID | 9824953 |
| InChIKey | QFOPFGRPNPCPBX-UHFFFAOYSA-N |
| Smiles | Cl.CC(C)(CC1=CNC2=CC=C(Cl)C=C12)NCCOC1=C(OCC2CC2)C=CC=C1 |
Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.
AllTocrisproductsareintendedforlaboratoryresearchuseonly.
SolubilityData
| Solvent | MaxConc.mg/mL | MaxConc.mM | |
|---|---|---|---|
| Solubility | |||
| DMSO | 22.47 | 50 | |
| ethanol | 4.49 | 10 |
PreparingStockSolutions
Thefollowingdataisbasedontheproductmolecularweight449.42.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.
| Concentration/SolventVolume/Mass | 1mg | 5mg | 10mg |
|---|---|---|---|
| 1mM | 2.23mL | 11.13mL | 22.25mL |
| 5mM | 0.45mL | 2.23mL | 4.45mL |
| 10mM | 0.22mL | 1.11mL | 2.23mL |
| 50mM | 0.04mL | 0.22mL | 0.45mL |
MolarityCalculator
ReconstitutionCalculator
DilutionCalculator
ProductDatasheets
© 2005- 苏州蚂蚁淘生物科技有限公司 版权所有。
苏ICP备17049038号-11
苏公网安备 32059002001627号
声明：本网站部分产品受外界条件影响（包含但不限于进口国出口国政策限制等因素），无法提供销售服务，下单后，会由客服人员联系厂家确认后另行通知。部分危险品无法清关，请勿下单
我要提问
您的问题将推送给已购用户，TA们将会为你解答。