BiologicalActivity
Selectiveσ1receptoragonist(IC50=17.4nM).Exhibitsselectivityforσ1overσ2receptors.InhibitsangiotensinII-inducedcardiomyocytehypertrophyinvitroandattenuatesmyocardialhypertrophyinvivo.Enhancesbrainplasticityandsensorimotorfunctioninaratmodelofexperimentalstroke.
CompoundLibraries
SA4503dihydrochlorideisalsoofferedaspartoftheTocriscreenPlus.FindoutmoreaboutcompoundlibrariesavailablefromTocris.
TechnicalData
| M.Wt | 441.43 |
| Formula | C23H32N2O2.2HCl |
| Storage | DesiccateatRT |
| Purity | ≥98%(HPLC) |
| CASNumber | 165377-44-6 |
| PubChemID | 9954941 |
| InChIKey | XWOXAKBQEMQMFH-UHFFFAOYSA-N |
| Smiles | COC1=C(OC)C=CC(CCN2CCN(CCCC3=CC=CC=C3)CC2)=C1.Cl.Cl |
Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.
AllTocrisproductsareintendedforlaboratoryresearchuseonly.
SolubilityData
| Solvent | MaxConc.mg/mL | MaxConc.mM | |
|---|---|---|---|
| Solubility | |||
| DMSO | 8.83 | 20 | |
| water | 44.14 | 100 |
PreparingStockSolutions
Thefollowingdataisbasedontheproductmolecularweight441.43.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.
| Concentration/SolventVolume/Mass | 1mg | 5mg | 10mg |
|---|---|---|---|
| 1mM | 2.27mL | 11.33mL | 22.65mL |
| 5mM | 0.45mL | 2.27mL | 4.53mL |
| 10mM | 0.23mL | 1.13mL | 2.27mL |
| 50mM | 0.05mL | 0.23mL | 0.45mL |
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