BiologicalActivity
Potentandselectivenociceptinopioidreceptor(NOP)agonist(EC50valuesare12,693,683and8071nM,andKivaluesare0.3,65,131and2854nMatNOP,μ-,κ-andδ-opioidreceptorsrespectively).Exhibitsanxiolytic-likeactivityatdosesthathavenoeffectonovertbehaviorssuchaslocomotioninvivo.Orallyactive.
CompoundLibraries
SCH221510isalsoofferedaspartoftheTocriscreenPlus.FindoutmoreaboutcompoundlibrariesavailablefromTocris.
TechnicalData
| M.Wt | 397.55 |
| Formula | C28H31NO |
| Storage | StoreatRT |
| Purity | ≥99%(HPLC) |
| CASNumber | 322473-89-2 |
| PubChemID | 9887077 |
| InChIKey | LOSJNRBXNQTUNT-UHFFFAOYSA-N |
| Smiles | OC1(C2=CC=CC=C2)CC3N(C(C5=CC=CC=C5C)C4=C(C)C=CC=C4)C(CC3)C1 |
Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.
AllTocrisproductsareintendedforlaboratoryresearchuseonly.
SolubilityData
| Solvent | MaxConc.mg/mL | MaxConc.mM | |
|---|---|---|---|
| Solubility | |||
| DMSO | 39.76 | 100 |
PreparingStockSolutions
Thefollowingdataisbasedontheproductmolecularweight397.55.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.
| Concentration/SolventVolume/Mass | 1mg | 5mg | 10mg |
|---|---|---|---|
| 1mM | 2.52mL | 12.58mL | 25.15mL |
| 5mM | 0.5mL | 2.52mL | 5.03mL |
| 10mM | 0.25mL | 1.26mL | 2.52mL |
| 50mM | 0.05mL | 0.25mL | 0.5mL |
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