BiologicalActivity
PotentandselectivecannABInoidCB1receptorantagonist(Ki=1.98nM).AlsoactsasaninverseagonistreversingadenylylcyclaseinhibitionbyWIN55,212-2(Cat.No.1038)(IC50=48nM).DisplaysnoactivityatCB2receptors.Reducesfoodintakeandbodyweightinorallydosednon-obeseWistarrats.
TechnicalData
| M.Wt | 500.25 |
| Formula | C22H21Cl3N4O.HCl |
| Storage | DesiccateatRT |
| Purity | ≥99%(HPLC) |
| CASNumber | 158681-13-1 |
| PubChemID | 104849 |
| InChIKey | REOYOKXLUFHOBV-UHFFFAOYSA-N |
| Smiles | O=C(NN4CCCCC4)C1=NN(C3=CC=C(Cl)C=C3Cl)C(C2=CC=C(Cl)C=C2)=C1C.Cl |
Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.
AllTocrisproductsareintendedforlaboratoryresearchuseonly.
SolubilityData
| Solvent | MaxConc.mg/mL | MaxConc.mM | |
|---|---|---|---|
| Solubility | |||
| DMSO | 50.02 | 100 |
PreparingStockSolutions
Thefollowingdataisbasedontheproductmolecularweight500.25.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.
| Concentration/SolventVolume/Mass | 1mg | 5mg | 10mg |
|---|---|---|---|
| 1mM | 2mL | 10mL | 19.99mL |
| 5mM | 0.4mL | 2mL | 4mL |
| 10mM | 0.2mL | 1mL | 2mL |
| 50mM | 0.04mL | 0.2mL | 0.4mL |
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