进口试剂Tocris直采 TOCRIS 4372-10MG,Tocris/TC-G 1008/5355/50/50 mg,受体,生物分子,生化试剂,,Tocris Bioscience蚂蚁淘商城

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Tocris/TC-G 1008/5355/50/50 mg

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Tocris

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5355/50

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4000-520-616

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Description:PotentandselectiveGPR39agoNIST

ChemicalName:N-[3-Chloro-4-[[[2-(methylamino)-6-(2-pyridinyl)-4-pyrimidinyl]amino]methyl]phenyl]methanesulfonamide

Purity:≥98%(HPLC)

BIOLOGicalActivityTechnicalDataSolubilityCalculatorsDatasheetsReferences

BiologicalActivity

PotentandselectiveGPR39agonist(EC₅₀valuesare0.4and0.8nMforratandhumanreceptorsrespectively).Selectiveoverapanelofkinases(IC₅₀s>10μM)anddisplaysminimalbindingaffinityforghrelinandneurotensin-1receptors(IC₅₀s>30μM).IncreasesGLP-1levelsinvitroandinvivo.Orallybioavailable.

CompoundLibraries

TC-G1008isalsoofferedaspartoftheTocriscreenPlus.FindoutmoreaboutcompoundlibrariesavailablefromTocris.

TechnicalData

M.Wt	418.9
Formula	C₁₈H₁₉ClN₆O₂S
Storage	Storeat+4°C
Purity	≥98%(HPLC)
CASNumber	1621175-65-2
PubChemID	91826086
InChIKey	DRSZMILOMUPIBJ-UHFFFAOYSA-N
Smiles	CNC1=NC(NCC2=C(Cl)C=C(NS(C)(=O)=O)C=C2)=CC(C3=NC=CC=C3)=N1

Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.

AllTocrisproductsareintendedforlaboratoryresearchuseonly.

SolubilityData

	Solvent	MaxConc.mg/mL	MaxConc.mM
Solubility
Solubility	DMSO	41.89	100

PreparingStockSolutions

Thefollowingdataisbasedontheproductmolecularweight418.9.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.

Concentration/SolventVolume/Mass	1mg	5mg	10mg
1mM	2.39mL	11.94mL	23.87mL
5mM	0.48mL	2.39mL	4.77mL
10mM	0.24mL	1.19mL	2.39mL
50mM	0.05mL	0.24mL	0.48mL

ProductDatasheets

CertificateofAnalysis/ProductDatasheet

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BiologicalActivity

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PreparingStockSolutions

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