BiologicalActivity
Potentandselectivenociceptin/orphaninFQ(NOP)receptorantagonist(pA2=7.75).DisplaysselectivityforNOPreceptorsoverclassicalopioidreceptors(pKivaluesare8.65,6.60,6.14and<5forNOP,μ-,κ-,andδ-opioidreceptorsrespectively).AttenuatesmotordeficitsinaratmodelofParkinson'sDisease.Activeinvivo.
CompoundLibraries
Trap101isalsoofferedaspartoftheTocriscreenPlus.FindoutmoreaboutcompoundlibrariesavailablefromTocris.
TechnicalData
| M.Wt | 434.02 |
| Formula | C24H35N3O2.HCl |
| Storage | Storeat+4°C |
| Purity | ≥98%(HPLC) |
| CASNumber | 1216621-00-9 |
| PubChemID | 56972178 |
| InChIKey | YEVMLMQAMCKVSC-UHFFFAOYSA-N |
| Smiles | Cl.CCN1C(=O)N(C2=CC=CC=C12)C1=C(CO)CN(CC2CCCCCCC2)CC1 |
Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.
AllTocrisproductsareintendedforlaboratoryresearchuseonly.
SolubilityData
| Solvent | MaxConc.mg/mL | MaxConc.mM | |
|---|---|---|---|
| Solubility | |||
| DMSO | 21.7 | 50 |
PreparingStockSolutions
Thefollowingdataisbasedontheproductmolecularweight434.02.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.
| Concentration/SolventVolume/Mass | 1mg | 5mg | 10mg |
|---|---|---|---|
| 1mM | 2.3mL | 11.52mL | 23.04mL |
| 5mM | 0.46mL | 2.3mL | 4.61mL |
| 10mM | 0.23mL | 1.15mL | 2.3mL |
| 50mM | 0.05mL | 0.23mL | 0.46mL |
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