BiologicalActivity
SelectivehistamineH4receptoragonist;displays50-foldselectivityfortheratH4receptorovertheH3subtype(pKivaluesare5.75and7.46forratH3andH4receptorsrespectively).AlsoexhibitsaffinityforthehumanH4receptor(pKi=8.22).
CompoundLibraries
VUF10460isalsoofferedaspartoftheTocriscreenPlus.FindoutmoreaboutcompoundlibrariesavailablefromTocris.
TechnicalData
| M.Wt | 269.34 |
| Formula | C15H19N5 |
| Storage | Storeat-20°C |
| Purity | ≥98%(HPLC) |
| CASNumber | 1028327-66-3 |
| PubChemID | 25129523 |
| InChIKey | NIJGWJIOMPHDBP-UHFFFAOYSA-N |
| Smiles | NC1=NC(C2=CC=CC=C2)=CC(N3CCN(C)CC3)=N1 |
Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.
AllTocrisproductsareintendedforlaboratoryresearchuseonly.
SolubilityData
| Solvent | MaxConc.mg/mL | MaxConc.mM | |
|---|---|---|---|
| Solubility | |||
| 2eq.HCl | 26.93 | 100 | |
| DMSO | 26.93 | 100 | |
| ethanol | 26.93 | 100 |
PreparingStockSolutions
Thefollowingdataisbasedontheproductmolecularweight269.34.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.
| Concentration/SolventVolume/Mass | 1mg | 5mg | 10mg |
|---|---|---|---|
| 1mM | 3.71mL | 18.56mL | 37.13mL |
| 5mM | 0.74mL | 3.71mL | 7.43mL |
| 10mM | 0.37mL | 1.86mL | 3.71mL |
| 50mM | 0.07mL | 0.37mL | 0.74mL |
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