BiologicalActivity
Potent,selectiveplatelet-activatingfactor(PAF)receptorantagonist(Ki=16.3nM).Displaysanti-inflammatory,antiangiogenicandanticanceractivity.InhibitsgrowthandproliferationofMCF-7breastcancercells.
CompoundLibraries
WEB2086isalsoofferedaspartoftheTocriscreenPlus.FindoutmoreaboutcompoundlibrariesavailablefromTocris.
TechnicalData
| M.Wt | 455.96 |
| Formula | C22H22N5O2SCl |
| Storage | Desiccateat+4°C |
| Purity | ≥99%(HPLC) |
| CASNumber | 105219-56-5 |
| PubChemID | 65889 |
| InChIKey | JGPJQFOROWSRRS-UHFFFAOYSA-N |
| Smiles | CC1=NN=C2CN=C(C3=C(SC(CCC(=O)N4CCOCC4)=C3)N12)C1=CC=CC=C1Cl |
Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.
AllTocrisproductsareintendedforlaboratoryresearchuseonly.
SolubilityData
| Solvent | MaxConc.mg/mL | MaxConc.mM | |
|---|---|---|---|
| Solubility | |||
| DMSO | 45.6 | 100 | |
| ethanol | 45.6 | 100mMwithgentlewarming |
PreparingStockSolutions
Thefollowingdataisbasedontheproductmolecularweight455.96.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.
| Concentration/SolventVolume/Mass | 1mg | 5mg | 10mg |
|---|---|---|---|
| 1mM | 2.19mL | 10.97mL | 21.93mL |
| 5mM | 0.44mL | 2.19mL | 4.39mL |
| 10mM | 0.22mL | 1.1mL | 2.19mL |
| 50mM | 0.04mL | 0.22mL | 0.44mL |
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