BiologicalActivity
PotentdopamineD4receptorpartialagonist(EC50=12.4nM;61%efficacyvs.dopamine).HasnoagonistactivityatD2receptors(EC50>10μM).Selectiveinratsinvivo;producespenileerectionfollowingi.c.v.administration;increasesintracavernosalpressureandpotentiatestheproerectileeffectsofsildenafilfollowings.c.administration.Displaysminimalsideeffects.
TechnicalData
| M.Wt | 402.75 |
| Formula | C17H19N5.3HCl |
| Storage | Desiccateat+4°C |
| Purity | ≥99%(HPLC) |
| CASNumber | 587870-77-7 |
| PubChemID | 16759165 |
| InChIKey | AZFUVPBLKQGSRI-UHFFFAOYSA-N |
| Smiles | Cl.Cl.Cl.C(N1CCN(CC1)C1=NC=CC=C1)C1=NC2=CC=CC=C2N1 |
Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.
AllTocrisproductsareintendedforlaboratoryresearchuseonly.
SolubilityData
| Solvent | MaxConc.mg/mL | MaxConc.mM | |
|---|---|---|---|
| Solubility | |||
| water | 40.27 | 100 |
PreparingStockSolutions
Thefollowingdataisbasedontheproductmolecularweight402.75.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.
| Concentration/SolventVolume/Mass | 1mg | 5mg | 10mg |
|---|---|---|---|
| 1mM | 2.48mL | 12.41mL | 24.83mL |
| 5mM | 0.5mL | 2.48mL | 4.97mL |
| 10mM | 0.25mL | 1.24mL | 2.48mL |
| 50mM | 0.05mL | 0.25mL | 0.5mL |
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