Tocris公司代理生物计划 Tocris Bioscience授权代理商，正品,Tocris/HC 067047/4100/50/50 mg,信号通路,细胞研究,细胞相关,,Tocris Bioscience蚂蚁淘商城

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Tocris/HC 067047/4100/50/50 mg

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Tocris

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4100/50

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Description:PotentandselectiveTRPV4antagoNIST

ChemicalName:2-Methyl-1-[3-(4-morpholinyl)propyl]-5-phenyl-N-[3-(trifluoromethyl)phenyl]-1H-pyrrole-3-carboxamide

Purity:≥99%(HPLC)

BIOLOGicalActivityTechnicalDataSolubilityCalculatorsDatasheetsReferences

BiologicalActivity

PotentandselectiveTRPV4antagonist.ReversIBLyinhibitscurrentsthroughmouse,humanandratTRPV4orthologs(IC₅₀valuesare17,48and133nMrespectively).AlsoinhibitstheendogenousTRPV4-mediatedresponseto4α-PDH(IC₅₀=22nM).SelectiveforTRPV4overTRPV1,TRPV2,TRPV3andTRPM8channels.

TechnicalData

M.Wt	471.51
Formula	C₂₆H₂₈F₃N₃O₂
Storage	Storeat+4°C
Purity	≥99%(HPLC)
CASNumber	883031-03-6
PubChemID	2742550
InChIKey	NCZYSQOTAYFTNM-UHFFFAOYSA-N
Smiles	CC1=C(C(NC4=CC(C(F)(F)F)=CC=C4)=O)C=C(C3=CC=CC=C3)N1CCCN2CCOCC2

Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.

AllTocrisproductsareintendedforlaboratoryresearchuseonly.

SolubilityData

	Solvent	MaxConc.mg/mL	MaxConc.mM
Solubility
	DMSO	47.15	100
	ethanol	11.79	25

PreparingStockSolutions

Thefollowingdataisbasedontheproductmolecularweight471.51.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.

Concentration/SolventVolume/Mass	1mg	5mg	10mg
1mM	2.12mL	10.6mL	21.21mL
5mM	0.42mL	2.12mL	4.24mL
10mM	0.21mL	1.06mL	2.12mL
50mM	0.04mL	0.21mL	0.42mL

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