Description:
Description:Phosphodiesterases(PDEs)playanimportantroleindynamicregulationofcAMPandcGMPsignaling.PDE7Aiswidelyexpressedinvarioustissuesincludingskeletalmuscle,Tlymphocytes,brainandpancreasandplaysandimportantroleintheregulationofosteoblasticdifferentiation.ThePDE7AAssayKitisdesignedforidentificationofPDE7Ainhibitorsusingfluorescencepolarization.TheassayisbasedonthebindingofafluorescentnucleotidemonophosphategeneratedbyPDE7Atothebindingagent.ThePDE7Ainhibitorscreeningassaykitcomesinaconvenient96-wellformat,includingpurifiedPDE7Aenzyme,fluorescentlylabeledPDE7Asubstrate(cAMP),bindingagent,andPDEassaybufferfor100enzymereactions.ThekeytothePDE7AAssayKitisthespecificbindingagent.Usingthiskit,onlytwosimplestepsonamicrotiterplatearerequiredforPDE7Areactions.First,thefluorescentlylabeledcAMPisincubatedwithasamplecontainingPDE7Afor1hour.Second,abindingagentisaddedtothereactionmixtoproduceachangeinfluorescentpolarizationthatcanthenbemeasuredusingafluorescencereader.Format:assaykit
ScientificCategory:PDE
AdditionalInformation:
| Name | PDE7AAssayKit |
|---|---|
| RelatedProductNames | PDE,phosphodiesterase,screening,inhibitors,PDE7A |
| Format | AssayKit |
| Storage | Mixedstorage |
| IntendedUse | ResearchUseOnly |

