BiologicalActivity
Metabolicallystableanandamideuptakeinhibitor(IC50=2.1-2.5μM)andfattyacidamidehydrolase(FAAH)inhibitor(Ki=3.18μM).InhibitsN-arachidonylethanolamine(AEA)accumulation(IC50=24μM)andhydrolysis(Ki=3μM),andinhibitsN-palmitoylethanolamine(PEA)hydrolysis(IC50=36μM)incerebellargranuleneurons.Alsoactsasanon-selectivecannABInoidreceptorpartialagonist(EC50valuesare189and271nMatCB2andCB1receptorsrespectively).
TechnicalData
| M.Wt | 409.6 |
| Formula | C27H39NO2 |
| Storage | Storeat-20°C |
| Purity | ≥98%(HPLC) |
| CASNumber | 251908-92-6 |
| PubChemID | 10364179 |
| InChIKey | XCWBOAHOJHPWLA-DOFZRALJSA-N |
| Smiles | CCCCCC=C/CC=C/C/C=CC/C=CCCCCNC(C1=CC=C(O)C=C1)=O |
Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.
AllTocrisproductsareintendedforlaboratoryresearchuseonly.
SolubilityData
| Solubility | Solubleinethanol(suppliedpre-dissolvedinanhydrousethanol,10mg/ml) |
PreparingStockSolutions
Thefollowingdataisbasedontheproductmolecularweight409.6.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.
| Concentration/SolventVolume/Mass | 1mg | 5mg | 10mg |
|---|---|---|---|
| 1mM | 2.44mL | 12.21mL | 24.41mL |
| 5mM | 0.49mL | 2.44mL | 4.88mL |
| 10mM | 0.24mL | 1.22mL | 2.44mL |
| 50mM | 0.05mL | 0.24mL | 0.49mL |
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