Tocris美元价/进货价 Tocris信号通路抑制剂,Tocris/AR-C155858/4960/1/1 mg,转运体,生物分子,生化试剂,,Tocris Bioscience蚂蚁淘商城

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Tocris/AR-C155858/4960/1/1 mg

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Tocris

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4960/1

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4000-520-616

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Description:MCT1andMCT2inhibitor;inhibitsglycolysisincancercells

ChemicalName:6-[(3,5-Dimethyl-1H-pyrazol-4-yl)methyl]-5-[[(4S)-4-hydroxy-2-isoxazolidinyl]carbonyl]-3-methyl-1-(2-methylpropyl)thieno[2,3-d]pyrimidine-2,4(1H,3H)-dione

Purity:≥98%(HPLC)

BIOLOGicalActivityTechnicalDataSolubilityCalculatorsDatasheetsReferences

BiologicalActivity

Inhibitorofthemonocarboxylatetransporters(MCTs)MCT1andMCT2(K_ivaluesare2.3and<10nMrespectively).ExhibitsnoactivityatMCT4.BlocksproliferationofRajilymphomacellsinvitro.Inhibitsglycolysisandglutathionesynthesisincancercells.

LicensingInformation

SoldforresearchpurposesunderagreementfromAstraZenecaUKLimited

TechnicalData

M.Wt	461.53
Formula	C₂₁H₂₇N₅O₅S
Storage	Storeat-20°C
Purity	≥98%(HPLC)
CASNumber	496791-37-8
PubChemID	10226546
InChIKey	ISIVOJWVBJIOFM-ZDUSSCGKSA-N
Smiles	O=C(N4OC[C@@H](O)C4)C1=C(CC3=C(C)NN=C3C)SC(N2CC(C)C)=C1C(N(C)C2=O)=O

Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.

AllTocrisproductsareintendedforlaboratoryresearchuseonly.

SolubilityData

	Solvent	MaxConc.mg/mL	MaxConc.mM
Solubility
Solubility	DMSO	46.15	100

PreparingStockSolutions

Thefollowingdataisbasedontheproductmolecularweight461.53.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.

Concentration/SolventVolume/Mass	1mg	5mg	10mg
1mM	2.17mL	10.83mL	21.67mL
5mM	0.43mL	2.17mL	4.33mL
10mM	0.22mL	1.08mL	2.17mL
50mM	0.04mL	0.22mL	0.43mL

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BiologicalActivity

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