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protein kinase, membrane associated tyrosine/threonine 1 | WEE family | IUPHAR/BPS Guide to PHARMACOLOGY

  
  2025-05-07
  
Annotated and awaiting review. Please contact us if you can help with reviewing. Description: Structure of human Membrane-associated Tyrosine- and Threonine-specific cdc2-inhibitory kinase MYT1 (PKMYT1) Download all structure-activity data for this target as a CSV file 1. Davis MI, Hunt JP, Herrgard S, Ciceri P, Wodicka LM, Pallares G, Hocker M, Treiber DK, Zarrinkar PP.(2011)Comprehensive analysis of kinase inhibitor selectivity. 2. Rohe A, Erdmann F, Bäßler C, Wichapong K, Sippl W, Schmidt M.(2012)In vitro and in silico studies on substrate recognition and acceptance of human PKMYT1, a Cdk1 inhibitory kinase. 3. Wang Y, Li J, Booher RN, Kraker A, Lawrence T, Leopold WR, Sun Y.(2001)Radiosensitization of p53 mutant cells by PD0166285, a novel G(2) checkpoint abrogator. 4. Wodicka LM, Ciceri P, Davis MI, Hunt JP, Floyd M, Salerno S, Hua XH, Ford JM, Armstrong RC, Zarrinkar PP et al..(2010)Activation state-dependent binding of small molecule kinase inhibitors: structural insights from biochemistry. WEE family: protein kinase, membrane associated tyrosine/threonine 1. Last modified on 19/02/2015. Accessed on 18/05/2020. IUPHAR/BPS Guide to PHARMACOLOGY, http://www.guidetopharmacology.org/GRAC/ObjectDisplayForward?objectId=2167.

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