BiologicalActivity
Potent,reversibleinhibitoroffattyacidamidehydrolase(FAAH)(IC50valuesare28and100nMforhumanandratFAAHrespectively).Noncovalentinhibitor;displaysselectivityforFAAHovercannABInoid-relatedtargets(IC50>20μMforCB1,CB2andTRPV1).Activeinvivo.
CompoundLibraries
TC-F2isalsoofferedaspartoftheTocriscreenPlus.FindoutmoreaboutcompoundlibrariesavailablefromTocris.
TechnicalData
| M.Wt | 439.51 |
| Formula | C26H25N5O2 |
| Storage | StoreatRT |
| Purity | ≥99%(HPLC) |
| CASNumber | 1304778-15-1 |
| PubChemID | 25198728 |
| InChIKey | NXTBLPPTZRPJCA-IBGZPJMESA-N |
| Smiles | O=C(N(CC)C6=C5C=CC=C6)N5[C@H]1CCCN(C2=NC(C3=CC(C=CC=C4)=C4O3)=CC=N2)C1 |
Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.
AllTocrisproductsareintendedforlaboratoryresearchuseonly.
SolubilityData
| Solvent | MaxConc.mg/mL | MaxConc.mM | |
|---|---|---|---|
| Solubility | |||
| DMSO | 43.95 | 100 |
PreparingStockSolutions
Thefollowingdataisbasedontheproductmolecularweight439.51.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.
| Concentration/SolventVolume/Mass | 1mg | 5mg | 10mg |
|---|---|---|---|
| 1mM | 2.28mL | 11.38mL | 22.75mL |
| 5mM | 0.46mL | 2.28mL | 4.55mL |
| 10mM | 0.23mL | 1.14mL | 2.28mL |
| 50mM | 0.05mL | 0.23mL | 0.46mL |
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