BiologicalActivity
Potentandselectivefattyacidamidehydrolase(FAAH)inhibitor(IC50valuesare3and5nMinhumanliverandratbrain,respectively).Exhibitsnosignificantinhibitoryactivityagainstavarietyofreceptors,ionchannelsandenzymes,includinghumancannABInoidreceptorsandratmonoacylglycerollipase.Displaysantiallodynicandantihyperalgesicactivityinaninflammatorypainmodel.
CompoundLibraries
URB597isalsoofferedaspartoftheTocriscreenPlus.FindoutmoreaboutcompoundlibrariesavailablefromTocris.
TechnicalData
| M.Wt | 338.4 |
| Formula | C20H22N2O3 |
| Storage | Storeat+4°C |
| Purity | ≥99%(HPLC) |
| CASNumber | 546141-08-6 |
| PubChemID | 1383884 |
| InChIKey | ROFVXGGUISEHAM-UHFFFAOYSA-N |
| Smiles | NC(C1=CC(C2=CC=CC(OC(NC3CCCCC3)=O)=C2)=CC=C1)=O |
Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.
AllTocrisproductsareintendedforlaboratoryresearchuseonly.
SolubilityData
| Solvent | MaxConc.mg/mL | MaxConc.mM | |
|---|---|---|---|
| Solubility | |||
| DMSO | 16.92 | 50 |
PreparingStockSolutions
Thefollowingdataisbasedontheproductmolecularweight338.4.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.
| Concentration/SolventVolume/Mass | 1mg | 5mg | 10mg |
|---|---|---|---|
| 1mM | 2.96mL | 14.78mL | 29.55mL |
| 5mM | 0.59mL | 2.96mL | 5.91mL |
| 10mM | 0.3mL | 1.48mL | 2.96mL |
| 50mM | 0.06mL | 0.3mL | 0.59mL |
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ProductDatasheets
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