BiologicalActivity
Orallyactiveantihypertensiveagentwhichdisplaysawiderangeofactivitiesinvitroandinvivo.InhibitsL-,N-andT-typeCa2+channels.Alsoinhibitsaldosterone-inducedmineralocorticoidreceptoractivation.Exhibitscardioprotectiveandantiartheroscleroticeffects.
TechnicalData
| M.Wt | 542.02 |
| Formula | C28H31N3O6.HCl |
| Storage | DesiccateatRT |
| Purity | ≥99%(HPLC) |
| CASNumber | 91599-74-5 |
| PubChemID | 76968919 |
| InChIKey | SPMJXDRNJQIBTB-IMEZZWDRSA-N |
| Smiles | CC1=C(C(OC)=O)[C@@H]([C@]2=CC([N+]([O-])=O)=CC=C2)C(C(O[C@H]3CN(CC4=CC=CC=C4)CCC3)=O)=C(C)N1.CC5=C(C(OC)=O)[C@H]([C@]6=CC([N+]([O-])=O)=CC=C6)C(C(O[C@@H]7CN(CC8=CC=CC=C8)CCC7)=O)=C(C)N5.Cl.Cl |
Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.
AllTocrisproductsareintendedforlaboratoryresearchuseonly.
SolubilityData
| Solvent | MaxConc.mg/mL | MaxConc.mM | |
|---|---|---|---|
| Solubility | |||
| DMSO | 40.65 | 75 | |
| ethanol | 5.42 | 10 |
PreparingStockSolutions
Thefollowingdataisbasedontheproductmolecularweight542.02.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.
| Concentration/SolventVolume/Mass | 1mg | 5mg | 10mg |
|---|---|---|---|
| 1mM | 1.84mL | 9.22mL | 18.45mL |
| 5mM | 0.37mL | 1.84mL | 3.69mL |
| 10mM | 0.18mL | 0.92mL | 1.84mL |
| 50mM | 0.04mL | 0.18mL | 0.37mL |
MolarityCalculator
ReconstitutionCalculator
DilutionCalculator
ProductDatasheets
© 2005- 苏州蚂蚁淘生物科技有限公司 版权所有。
苏ICP备17049038号-11
苏公网安备 32059002001627号
声明：本网站部分产品受外界条件影响（包含但不限于进口国出口国政策限制等因素），无法提供销售服务，下单后，会由客服人员联系厂家确认后另行通知。部分危险品无法清关，请勿下单
我要提问
您的问题将推送给已购用户，TA们将会为你解答。