BiologicalActivity
Potent,selectiveandcompetitivebenzodiazepinereceptorantagonist(IC50valuesare0.4and0.7nMforinhibitionof[3H]-flunitrazepambindingtoratcerebellumandhippocampusrespectively).Similarinvivoprofiletoflumazenil(Ro15-1788,CatNo.1328);producesanxiogeniceffectsinsomebehavioraltestsandanxiolyticeffectsinothers.Orallyactive.
CompoundLibraries
ZK93426hydrochlorideisalsoofferedaspartoftheTocriscreenPlus.FindoutmoreaboutcompoundlibrariesavailablefromTocris.
TechnicalData
| M.Wt | 348.82 |
| Formula | C18H20N2O3.HCl |
| Storage | DesiccateatRT |
| Purity | ≥99%(HPLC) |
| CASNumber | 1216792-30-1 |
| PubChemID | 56972167 |
| InChIKey | RNQJDOYVHCISJU-UHFFFAOYSA-N |
| Smiles | Cl.CCOC(=O)C1=C(C)C2=C(NC3=C2C(OC(C)C)=CC=C3)C=N1 |
Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.
AllTocrisproductsareintendedforlaboratoryresearchuseonly.
SolubilityData
| Solvent | MaxConc.mg/mL | MaxConc.mM | |
|---|---|---|---|
| Solubility | |||
| DMSO | 17.44 | 50 | |
| water | 34.88 | 100 |
PreparingStockSolutions
Thefollowingdataisbasedontheproductmolecularweight348.82.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.
| Concentration/SolventVolume/Mass | 1mg | 5mg | 10mg |
|---|---|---|---|
| 1mM | 2.87mL | 14.33mL | 28.67mL |
| 5mM | 0.57mL | 2.87mL | 5.73mL |
| 10mM | 0.29mL | 1.43mL | 2.87mL |
| 50mM | 0.06mL | 0.29mL | 0.57mL |
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